Purpose
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SGX-523 is a selective Met inhibitor with IC50 of 4 nM, no activity to BRAFV599E, c-Raf, Abl and p38α. Phase 1.
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Characteristics
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Target: c-Met inhibitor, Raf inhibitor, Bcr-Abl inhibitor, p38 MAPK inhibitor Receptor: c-Met,B-Raf/C-Raf/Abl/p38α
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Purification
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All the products are sent with COA, HPLC and NMR inspection report to guarantee the quality.
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Purity
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97?% +
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Formula
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C18H13N7S
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Solubility
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5 mM in DMSO
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