產(chǎn)品詳情
所在位置: 首頁> 產(chǎn)品目錄> 試劑>
  • 產(chǎn)品名稱:Prasugrel

  • 產(chǎn)品型號:
  • 產(chǎn)品廠商:TargetMol
  • 產(chǎn)品文檔:
你添加了1件商品 查看購物車
簡單介紹:
Prasugrel
詳情介紹:
Purpose Prasugrel, a thienopyridine derivative, is a platelet activation and aggregation inhibitor structurally and pharmacologically related to clopidogrel and ticlopidine. Similar to clopidogrel, prasugrel is a prodrug that requires enzymatic transformation in the liver to its active metabolite, R-138727. R-138727 irreversibly binds to P2Y12 type ADP receptors on platelets thus preventing activation of the GPIIb/IIIa receptor complex. As a result, inhibition of ADP-mediated platelet activation and aggregation occurs. Prasugrel was developed by Daiichi Sankyo Co. and is currently marketed in the United States and Canada in cooperation with Eli Lilly and Company for acute coronary syndromes planned for percutaneous coronary intervention (PCI). FDA approved in 2009.
Characteristics Tradename: EFFIENT
Source of Compound: synthetic
Target: P2 Receptor antagonist
Receptor: Cocaine esterase, P2Y Receptor
Status: USAN, INN
Purification All the products are sent with COA, HPLC and NMR inspection report to guarantee the quality.
Purity 99?%
Formula C20H20FNO3S
Solubility In water, 20.28 mg/L
Molecular Weight 373.44 g/mol
CAS-No 150322-43-3
Application Notes Optimal working dilution should be determined by the investigator.
Restrictions For Research Use only
Format Solid
Storage -20 °C
Storage Comment For the majority of compounds, they could be dissolved in DMSO or other organic solvent.
Their stock solution can be stored at -20°C for up to 3 months and aliquoted for sampling convenience.
Several freeze/thaw cycles should not damage the activity of our small molecule products.
However, in many instances the aqueous solutions of some compounds need to be made fresh and cannot be stored. For these compounds, their solution should be prepared just before use and stored no longer than 24 hours.
Expiry Date 24 months