Purpose
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LY364947 is a potent ATP-competitive inhibitor of TGFβR-I with IC50 of 59 nM in a cell-free assay, shows 7-fold selectivity over TGFβR-II.
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Characteristics
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Target: TGF-beta/Smad inhibitor, CK inhibitor Receptor: TGFβRI,RIPK2,CK1δ,TGFβRII,MLK-7K
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Purification
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All the products are sent with COA, HPLC and NMR inspection report to guarantee the quality.
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Purity
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98?%
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Formula
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C17H12N4
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Solubility
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10 mM in DMSO
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