產(chǎn)品詳情
  • 產(chǎn)品名稱:Apremilast

  • 產(chǎn)品型號(hào):
  • 產(chǎn)品廠商:Biovision
  • 產(chǎn)品文檔:
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Apremilast
詳情介紹:
Characteristics Apremilast is a potent PDE4 (phosphodiesterase 4) inhibitor (IC50= 74 nM). It reduces TNF-alpha production in human synovial cells and significantly suppresses experimental arthritis.
Purity ≥ 98?% by HPLC
Chemical Name N-{2-[(1S)-1-(3-Ethoxy-4-methoxyphenyl)-2-(methylsulfonyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}acetamide
Formula C??H??N?O?S
Permeability Cell-permeable
Molecular Weight 460.5 g/mol
CAS-No 608141-41-9
Restrictions For Research Use only
Format Solid
Handling Advice Protect from air and moisture
Storage -20 °C
Expiry Date 36 months
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 image for Apremilast (ABIN1685730) Apremilast