Characteristics
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Cell-permeable. A potent, selective and ATP-competitive inhibitor of PI 3-kinase beta (IC50 = 5 nM for p110beta). Inhibits other PI3K isoforms at higher concentrations (IC50 = 0.1 μM for p110delta, 5 μM for p110beta, and 3.5 μM for p110alpha).
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