Purpose
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UNC1999 is a potent, orally bioavailable and selective inhibitor of EZH2 and EZH1 with IC50 of 2 nM and 45 nM in cell-free assays, respectively, showing >1000-fold selectivity over a broad range of epigenetic and non-epigenetic targets.
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Characteristics
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Target: Histone Methyltransferase inhibitor Receptor: EZH2,EZH1 Status: Undetermined activity
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Purification
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All the products are sent with COA, HPLC and NMR inspection report to guarantee the quality.
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Purity
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100?%
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Formula
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C33H43N7O2
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Solubility
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DMSO 100 mg/Ml,Ethanol 100 mg/mL,
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