Purpose
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PIK-75 is a p110α inhibitor with IC50 of 5.8 nM (200-fold more potently than p110β), isoform-specific mutants at Ser773, and also potently inhibits DNA-PK with IC50 of 2 nM in cell-free assays.
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Characteristics
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Target: PI3K inhibitor, DNA-PK inhibitor Receptor: DNA-PK,p110α,p110γ,p110δ,p110β
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Purification
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All the products are sent with COA, HPLC and NMR inspection report to guarantee the quality.
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Purity
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97?% +
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Formula
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C16H14BrN5O4S.HCl
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Solubility
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10 mM in DMSO
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